Found 5 results
Author Title [ Type(Desc)] Year
Filters: Author is Scapozza, Leonardo  [Clear All Filters]
Journal Article
M. Ceccon, Mologni, L., Bisson, W. H., Scapozza, L., and Gambacorti-Passerini, C., Crizotinib-resistant NPM-ALK mutants confer differential sensitivity to unrelated Alk inhibitors, Molecular Cancer Research, vol. 11, pp. 122–132, 2013.
T. Wang, Bisson, W. H., Mäser, P., Scapozza, L., and Picard, D., Differences in conformational dynamics between Plasmodium falciparum and human Hsp90 orthologues enable the structure-based discovery of pathogen-selective inhibitors, Journal of medicinal chemistry, vol. 57, pp. 2524–2535, 2014.
W. H. Bisson, Westera, G., P Schubiger, A., and Scapozza, L., Homology modeling and dynamics of the extracellular domain of rat and human neuronal nicotinic acetylcholine receptor subtypes $\alpha$4$\beta$2 and $\alpha$7, Journal of molecular modeling, vol. 14, pp. 891–899, 2008.
W. H. Bisson, Scapozza, L., Westera, G., Mu, L., and Schubiger, P. A., Ligand selectivity for the acetylcholine binding site of the rat $\alpha$4$\beta$2 and $\alpha$3$\beta$4 nicotinic subtypes investigated by molecular docking, Journal of medicinal chemistry, vol. 48, pp. 5123–5130, 2005.
S. Tardy, Orsato, A., Mologni, L., Bisson, W. H., Donadoni, C., Gambacorti-Passerini, C., Scapozza, L., Gueyrard, D., and Goekjian, P. G., Synthesis and biological evaluation of benzo [4, 5] imidazo [1, 2-c] pyrimidine and benzo [4, 5] imidazo [1, 2-a] pyrazine derivatives as anaplastic lymphoma kinase inhibitors, Bioorganic & medicinal chemistry, vol. 22, pp. 1303–1312, 2014.